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(19)

(11)

2 446 167

(13)

(51)

IPC

C07D401/12(2006-01-01)

C07D409/04(2006-01-01)

C07D213/74(2006-01-01)

C07D213/40(2006-01-01)

C07D213/64(2006-01-01)

C07D295/12(2006-01-01)

C07D311/08(2006-01-01)

A61K31/444(2006-01-01)

(21) (22)

Application

2008119415/04, 2006-10-19

(24)

Start date

2006-10-19

(22)

Actual filing date

2006-10-19

(45)

Published

2012-03-27

(72)

Inventor

Li ChzhivuRe Khen ChulFrank RobertBarenberg GregorDe-Vri ZhanKristof TomasSonders Derek DzhonShine KlausZundermann Bernd

(73)

Holder

Grjunental' Gmbkh

NEW COMPOUNDS - VANILLOID RECEPTOR LIGANDS AND USE OF SUCH COMPOUNDS FOR PREPARING DRUGS Russian patent published in 2012 - IPC C07D401/12 C07D409/04 C07D213/74 C07D213/40 C07D213/64 C07D295/12 C07D311/08 A61K31/444

Abstract RU 2446167 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to a new compound of formula A

the radicals R¹, R², R³, R⁴, R⁵, R²⁵, R²⁶, U, T, W, V, Y are those as specified in clause 1 of the patent claim. Also, the invention refers to a method for preparing the compound of formula A, the drug based on this compound applied for treating disorders or diseases which are at least partially mediated by vanilloid receptor VR1 /NRPV1, as well as use of this compound for preparing the drug.

EFFECT: there are prepared and described new compounds which can be effective in treating diseases which are at least partially mediated by vanilloid receptor VR1 /NRPV1.

43 cl, 367 ex, 4 tbl

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RU 2 446 167 C2

Authors

Li Chzhivu

Re Khen Chul

Frank Robert

Barenberg Gregor

De-Vri Zhan

Kristof Tomas

Sonders Derek Dzhon

Shine Klaus

Zundermann Bernd

Dates

2012-03-27—Published

2006-10-19—Filed