FIELD: chemistry.
SUBSTANCE: claim describes novel vinylogous acid derivatives of formula 
, in which ring A is as defined in claim 1, R1 denotes hydrogen, C1-C6-alkyl or -NR'R", -( C0-C6-alkylene)-NR'R'', where R' and R" are independently selected from a group comprising hydrogen, C1-C6-alkyl, formyl, C1-C6-alkylcarbonyl; R2, R2' and R2" independently denote hydrogen, halogen, C1-C6-alkyl or C1-C6-alkoxy group; R3 denotes phenyl; R4 denotes hydrogen, C1-C6-alkyl, optionally substituted phenyl or phenyl- C1-C6-alkyl, R5 denotes hydrogen or C1-C6-alkyl; as well as physiologically acceptable salts thereof.
EFFECT: compounds inhibit chymase and can be used as medicinal agents.
15 cl, 27 ex
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