INSECTICIDAL ARYL PYRROLIDINES Russian patent published in 2013 - IPC C07D207/04 C07D401/04 C07D401/14 C07D403/10 A01N43/36 A01N43/40 

FIELD: chemistry.

SUBSTANCE: invention concerns novel aryl pyrrolidines of formula I:

, where X, which can be identical or different, denote halogen, halogen-C_1-6alkyl, NO₂, C_1-6alkyl, C_1-6alkoxy, CN, halogen-C_1-6alkoxy, C_1-6alkylthio, C_1-6alkylthionyl, C_1-6alkylsulphonyl, halogen- C_1-6alkylthio, halogen- C_1-6alkylthionyl, halogen- C_1-6alkylsulphonyl, OH, mercapto groups, NH₂, C_1-6alkylcarbonyl amino groups, halogen- C_1-6alkylcarbonyl-amino, C_1-6alkoxycarbonyl amino groups, halogen-C_1-6alkoxycarbonylamino; Y, which can be identical or different, denote halogen, halogen- C_1-6alkyl, NO₂, C_1-6alkyl, C_1-6alkoxy, CN, halogen- C_1-6alkoxy, C_1-6alkylthio, C_1-6alkylthionyl, C_1-6alkylsulphonyl, halogen- C_1-6alkylthio, halogen- C_1-6alkylthionyl, halogen- C_1-6alkylsulphonyl, hydroxyl groups, mercapto groups, NH₂, C_1-6alkylcarbonyl amino groups, halogen- C_1-6alkylcarbonyl amino, C_1-6alkoxycarbonyl amino groups, halogen- C_1-6alkoxycarbonyl amino; R denotes halogen- C_1-6alkyl; m equals 0, 1, 2, 3, 4, 5; n equals 1, 2, 3, 4; G denotes a group: , where R¹ and R² each independently denotes H, unsubstituted C_1-6alkyl, halogen- C_1-6alkyl, -CH₂R⁷;R³, R⁴ each independently denotes H; I equals 1, 2, 3; R⁵ denotes H; R⁶ denotes C_1-6alkylcarbonyl, a group: G6 - G8:

b where k³ equals 0; k⁴ equals 0; R⁷ denotes an unsubstituted 6-member heteroaryl with one N; A denotes C, N.

EFFECT: compounds exhibit insecticidal activity, which enables use thereof in insect and/or tick control method.

7 cl, 13 tbl, 8 ex