CYCLIC INDOLE-3-CARBOXAMIDE, PRODUCTION AND USE THEREOF AS THERAPEUTIC PREPARATIONS Russian patent published in 2013 - IPC C07D209/42 C07D403/12 C07D405/04 C07D409/04 A61K31/496 A61P9/12 

Abstract RU 2485102 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to cyclic indole-3-carboxamide of formula (I) or physiologically acceptable salts thereof of formula (I): wherein the values A, R, R10, R20, R30, R40, n, p and q are specified in clause 1 of the patent claim. A method for preparing them is described.

EFFECT: compounds have renin-inhibitory activity that allows using them for preparing a pharmaceutical composition and a drug preparation for treating the diseases associated with renin activity.

11 cl, 4 tbl, 127 ex

Similar patents RU2485102C2

Title Year Author Number
CYCLIC AZAINDOLE-3-CARBOXAMIDE, PRODUCTION AND USE THEREOF AS THERAPEUTIC PREPARATIONS 2009
  • Shtajnkhagen Khenning
  • Shajper Bodo
  • Matter Khans
  • Makkort Gari
RU2487874C2
CYCLIC (AZA)INDOLYSINCARBOXAMIDES, PREPARING AND USING THEM AS PHARMACEUTICAL AGENTS 2010
  • Shtajnkhagen Khenning
  • Shajper Bodo
  • Matter Khans
  • Makkort Gari
  • Bezhi Gijom
  • Gobervill' Paskal'
  • T'Er Beranzher
RU2539574C2
NOVEL DERIVATIVES OF IMIDAZOLIDINE, THEIR PREPARING, THEIR APPLICATION AND PHARMACEUTICAL PREPARATIONS CONTAINING THEREOF 1998
  • Vener Fol'Kmar
  • Shtil'Ts Khans Ul'Rikh
  • Shmidt Vol'Fgang
  • Zajffge Dirk
RU2213737C2
INHIBITORS OF FACTOR VIIA 2000
  • Klingler Otmar
  • Shudok Manfred
  • Tsoller Gerkhard
  • Khajnel'T Uve
  • Defossa Ehlizabet
  • Matter Khans
  • Safar Pavel
RU2248359C2
DERIVATIVES OF (THIO)UREA INHIBITING VIIa FACTOR, METHOD FOR THEIR PREPARING AND PHARMACEUTICAL COMPOSITION 2001
  • Klingler Otmar
  • Shudok Manfred
  • Nestler Khans-Peter
  • Matter Khans
  • Shrojder Kherman
RU2286337C2
NEW FIVE-MEMBER HETEROCYCLES, THEIR PREPARING, THEIR APPLYING AND PHARMACEUTICAL PREPARATIONS COMPRISING THEREOF 1998
  • Vener Fol'Kmar
  • Shtil'Ts Khans Ul'Rikh
  • Shmidt Vol'Fgang
  • Zajffge Dirk
RU2240326C2
FIVE-MEMBERED HETEROCYCLES AS INHIBITORS OF LEUKOCYTE ADHESION AND VLA-4 ANTAGONISTS 1997
  • Shtil'Ts Khans Ul'Rikh
  • Vener Fol'Kmar
  • Knolle Jokhen
  • Bartnik Ehkart
  • Khjul'S Kristof
RU2229296C2
SUBSTITUTED DERIVATIVES OF IMIDAZOLIDINE, METHOD FOR PREPARING AND PHARMACEUTICAL PREPARATION 1998
  • Vener Fol'Kmar
  • Shtil'Ts Khans Ul'Rikh
  • Shmidt Vol'Fgang
  • Zajffge Dirk
RU2239641C2
NOVEL DERIVATIVES OF IMIDAZOLIDINE, THEIR PREPARING AND USING AS VLA-4 ANTAGONIST 2002
  • Vener Fol'Kmar
  • Flor Shtefani
  • Blum Khorst
  • Rjutten Khartmut
  • Shtil'Ts Khans Ul'Rikh
RU2318815C2
SUBSTITUTED INDOLES 2000
  • Rittseler Olaf
  • Shtil'Ts Khans Ul'Rikh
  • Najses Bernkhard
  • Ene Gerkhard
  • Khabermann Jorg
RU2255087C2

RU 2 485 102 C2

Authors

Shtajnkhagen Khenning

Shajper Bodo

Matter Khans

Shtil'Ts Khans Ul'Rikh

Makkort Gari

Dates

2013-06-20Published

2009-01-17Filed