OCTAHYDROPYRROLO[3,4-b]PYRROLE DERIVATIVES (VERSIONS), METHOD OF OBTAINING OCTAHYDROPYRROLO[3,4-b]PYRROLE DERIVATIVES (VERSIONS), BASED ON THEM PHARMACEUTICAL COMPOSITION AND METHOD OF TREATING DISEASE OR IMPAIRMENT OF STATE OF ORGANISM, SENSITIVE TO MODULATION OF HISTAMINE-3 RECEPTOR ACTIVITY Russian patent published in 2013 - IPC C07D487/04 A61K31/407 

Abstract RU 2492172 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention relates to ocrahydropyrrolo[3,4-b]pyrrole derivatives of formula I: or their pharmaceutically acceptable salts, where values R1, R2a, R2b, R2c, R2d, R2e, R2f, R3a , R3b, R3c, R3d, Cy1, L2, Cy2 are given in item 1 of the formula. Method of their obtaining is described.

EFFECT: compounds can be used for treatment of organism therapeutically sensitive to binding of histamine-3 receptor.

47 cl, 22 dwg, 6 tbl, 87 ex

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RU 2 492 172 C2

Authors

Barns Dehvid M.

Blehk Lorens A.

Vittenberger Stiven Dzh.

Grehg Robert Dzh.

Kauehrt Marlon D.

Kolachkovski Lorens

Lou Sjaochun'

San Minkhua

Fiks Majkl G.

Khajt Ehntoni R.

Khenri Rodzher F.

Chan Sou-Tszehn'

Chzhan Dzheff G. Z.

Chzhao Chehn'

Chzhehn Go Chzhu

Shejkh Akhmad I.

Dates

2013-09-10Published

2007-02-16Filed