FIELD: chemistry.
SUBSTANCE: disclosed are compositions having sodium-dependent glucose cotransporter
(SGLT) inhibiting effect, having a structure given below, where values of radicals are given in the claim. Also disclosed is a method of treating or preventing a disease influenced by SGLT inhibition, where said disease is: type 1 sugar diabetes, type 2 sugar diabetes, hyperglycemia, diabetic complications, insulin resistance, metabolic syndrome (Syndrome X), hyperinsulinemia, hypertension, hyperuricemia, obesity, oedema, dyslipidemia, chronic heart failure or atherosclerosis.
EFFECT: invention also provides pharmaceutical compositions and methods for deuterium-enrichment of a diaryl methyl compound, having a structure given below, where values of radicals are given in the claim.
37 cl, 7 dwg, 6 tbl, 64 ex
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