COMPOSITIONS OF TELMISARTAN IN FORM OF NANOPARTICLES, AND METHOD FOR PREPARING THEM Russian patent published in 2014 - IPC A61K9/14 A61K31/4184 A61P9/12 

Abstract RU 2526914 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to pharmaceutics, namely to a stable pharmaceutical composition of nanostructured telmisartan for treating hypertension, containing nanostructured telmisartan having an average particle size less than approximately 600 nm, and at least one stabilising agent specified in a group of sodium dodecyl sulphate and polyvinyl pyrrolidone, wherein the composition in prepared in a continuous flow reactor, preferentially in a microfluidics continuous flow reactor, as well as to a method for preparing the composition and using it.

EFFECT: invention provides better physical-chemical characteristics and pharmacokinetics of the active principle.

11 cl, 9 ex, 3 tbl, 14 dwg

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RU 2 526 914 C2

Authors

Filipchei Genoveva

Ehtvesh Zhol'T

Pongrats Katalin

Darvash Ferents

Dates

2014-08-27Published

2010-06-18Filed