FIELD: chemistry.
SUBSTANCE: invention relates to a novel compound of formula I-1, characterised by effects of thrombolysis, accepting free radicals and directed action on thrombus. Compound is a three-component conjugate formed by conjugation of thrombolytic oligopeptide, free radical acceptor and a peptide with directed action on thromb/antithrombotic oligopeptide by binder link.
EFFECT: present invention also relates to a pharmaceutical composition containing compounds, wherein compounds form a nanospherical structure.
13 cl, 40 dwg, 21 tbl, 17 ex
Title | Year | Author | Number |
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NEW COMPOUNDS HAVING TRIPLE ACTIVITIES OF THROMBOLYSIS, ANTITHROMBOTIC AND RADICAL SCAVENGING, AND SYNTHESIS, NANO-STRUCTURE AND USE THEREOF | 2014 |
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Authors
Dates
2016-12-10—Published
2013-03-15—Filed