NOVEL COMPOUND WITH EFFECTS OF THROMBOLYSIS, ACCEPTING FREE RADICALS AND DIRECTED ACTION ON THROMBUS, AS WELL AS METHOD FOR PRODUCTION AND USE THEREOF Russian patent published in 2016 - IPC C07K7/06 C07K1/06 A61K38/08 A61K31/41 A61P7/02 A61P39/06 A61P9/10 

Abstract RU 2604193 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a novel compound of formula I-1, characterised by effects of thrombolysis, accepting free radicals and directed action on thrombus. Compound is a three-component conjugate formed by conjugation of thrombolytic oligopeptide, free radical acceptor and a peptide with directed action on thromb/antithrombotic oligopeptide by binder link.

EFFECT: present invention also relates to a pharmaceutical composition containing compounds, wherein compounds form a nanospherical structure.

13 cl, 40 dwg, 21 tbl, 17 ex

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RU 2 604 193 C2

Authors

Peng Shiqi

Zhao Ming

Jiang Xueyun

Dates

2016-12-10Published

2013-03-15Filed