FIELD: pharmacology.
SUBSTANCE: invention relates to 5-aryl-substituted 4-(5-nitrofuran-2-yl)pyrimidines , as well as a process for their preparation using intermediate compound. The resulting compounds (Ia-d and II) can be used to treat patients with diseases of the genitourinary system caused by Staphylococcus aureus or gonococci.
EFFECT: highly effective method for preparation of these compounds, which have a broad spectrum of antibacterial activity, is proposed.
3 cl, 2 tbl, 4 ex
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Authors
Dates
2017-07-31—Published
2016-08-19—Filed