CRYSTALLINE FORMS OF GRAPIPRANT Russian patent published in 2017 - IPC C07D471/04 A61K31/437 A61P29/00 

Abstract RU 2638931 C1

FIELD: pharmacology.

SUBSTANCE: invention relates to the crystalline form of grapiprant selected from the group consisting of Form X, Form X2, Form X3, Form F, Form K, Form L, Form M and Form N.

EFFECT: new crystalline form of grapiprant, as well as pharmaceutical compositions suitable for treatment of pain, inflammation, arthritis and cancer, and methods to obtain them.

8 cl, 13 tbl, 23 dwg, 12 ex

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RU 2 638 931 C1

Authors

Nyubold Tamara

Smit Melissa

Sikamp Kris

Venslou Robert

Lyu Sya

Dates

2017-12-19Published

2015-03-05Filed