Show metadata Hide metadata

(19)

(11)

2 640 579

(13)

(51)

IPC

C07D473/00(2006-01-01)

A61K31/52(2006-01-01)

A61P7/02(2006-01-01)

(21) (22)

Application

2017112242, 2017-04-10

(24)

Start date

2017-04-10

(22)

Actual filing date

2017-04-10

(45)

Published

2018-01-10

(72)

Inventor

Khaliullin Ferkat AdelzyanovichShabalina Yuliya ViktorovnaSamorodov Aleksandr VladimirovichKamilov Feliks KhusainovichMustafin Ilshat Ganievich

(73)

Holder

Khaliullin Ferkat Adelzyanovich

HYDROCHLORIDES OF 1-ALKYL-3-METHYL-8-PIPERAZINO-7-(TIETHANYL-3)XANTHINE SHOWING ANTITHROMBOTIC EFFECT BY BLOCKING GP IIb-IIIa PLATELETS RECEPTORS Russian patent published in 2018 - IPC C07D473/00 A61K31/52 A61P7/02

Abstract RU 2640579 C1

FIELD: pharmacology.

SUBSTANCE: invention relates to 1-alkyl-3-methyl-8-piperazino-7-(tiethanyl-3)xanthine hydrochlorides of the general formula: Ia-c, where R=CH₂-CH=CH₂ (Ia), C₃H₇-iso (Ib), C₅H₁₁-h (Ic).

EFFECT: increased antithrombotic effect by blocking the GP IIb-IIIa platelet receptors.

5 cl, 2 tbl, 5 ex

Similar patents RU2640579C1

Title	Year	Author	Number
MEANS SHOWING ANTITHROMBOTIC EFFECT BY BLOCKING GP IIb-IIIa PLATELETS RECEPTORS (VERSIONS)	2016	Khaliullin Ferkat Adelzyanovich Samorodov Aleksandr Vladimirovich Shabalina Yuliya Viktorovna Kamilov Feliks Khusainovich Mustafin Ilshat Ganievich Khalimov Almaz Radykovich	RU2643336C1
AGENT FOR TREATMENT AND PREVENTION OF THROMBOSIS	2017	Khaliullin Ferkat Adelzyanovich Samorodov Aleksandr Vladimirovich Shabalina Yuliya Viktorovna Kamilov Feliks Khusainovich	RU2662308C1
DERIVATIVES OF THIAETANE-CONTAINING 1-BUTYL-3-METHYLXANTHINES EXHIBITING ANTIOXIDANT ACTIVITY	2020	Khaliullin Ferkat Adelzyanovich Samorodov Aleksandr Vladimirovich Mamatov Zhekshen Kasenovich Bashirova Linara Irekovna Timirkhanova Galiya Amirovna Bashirov Ilnur Irekovich Amatova Nurzada Zhanyshevna	RU2740926C1
DERIVATIVES OF 3-METHYL-7-(THETANYL-3)-XANTHINE POSSESSING HEMORHEOLOGICAL ACTIVITY	2006	Khaliullin Ferkat Adel'Zjanovich Filipenko Julija Viktorovna Saitgalina Ajgul' Zakirovna Spasov Aleksandr Alekseevich Naumenko Ljudmila Vladimirovna	RU2316551C1
CYCLOHEXYL AMMONIUM SALT OF 2-[3-METHYL-7-(1,1-DIOXOTIETHANYL-3)-1-ETHYL XANTHENYL-8-TIO]ACETIC ACID, WHICH SHOWS ANTITHROMBOEMBOLIC ACTION	2012	Khaliullin Ferkat Adel'Zjanovich Murataev Danijar Zamirovich Shabalina Julija Viktorovna Kamilov Feliks Khusainovich Timirkhanova Galija Amirovna Samorodova Al'Bina Ildarovna	RU2504546C1
3-METHYL-8-PIPERAZINE-7-(THIETHANYL-3)-1-ETHYLXANTHINE HYDROCHLORIDE, EXHIBITING ANTIAGGREGANT AND DISAGGREGATION ACTIVITY	2009	Khaliullin Ferkat Adel'Zjanovich Shabalina Julija Viktorovna Timirkhanova Galija Amirovna Kamilov Feliks Khusainovich Samorodov Aleksandr Vladimirovich Sharafutdinov Ruslan Maratovich	RU2404181C1
2-BROMO-1-(THIETANYL-3)IMIDAZOLE-4,5-DICARBOXYLIC ACID DERIVATIVES EXHIBITING ANTIDEPRESSANT ACTIVITY	2014	Khaliullin Ferkat Adel'Zjanovich Nikitina Irina Leonidovna Valieva Anfisa Rifovna Miftakhova Al'Bina Fljurovna Magadeeva Gul'Naz Fatikhovna Ivanova Ol'Ga Aleksandrovna Alekhin Evgenij Konstantinovich	RU2537948C1
SALTS OF [3-METHYL-1-N-PROPYL-7-(1,1-DIOXOTHIETANYL-3)XANTHINYL-8-THIO]ACETIC ACID, EXHIBITING PROAGGREGANT ACTIVITY	2011	Kamilov Feliks Khusainovich Timirkhanova Galija Amirovna Samorodov Aleksandr Vladimirovich Khalimov Almaz Radykovich Khaliullin Ferkat Adel'Zjanovich Gubaeva Regina Amurovna Shabalina Julija Viktorovna	RU2459825C1
CYCLOHEXYLAMMONIUM SALT OF [3-METHYL-1-N-PROPYL-7-(1-OXOTHIETANYL-3)XANTHINYL-8-THIO]ACETIC ACID EXHIBITING ANTITHROMBOTIC ACTIVITY	2011	Khaliullin Ferkat Adel'Zjanovich Gubaeva Regina Amurovna Shabalina Julija Viktorovna Kamilov Feliks Khusainovich Timirkhanova Galija Amirovna Samorodov Aleksandr Vladimirovich	RU2459826C1
AGENT EXHIBITING ANTIAGGREGATORY ACTIVITY	2019	Urakov Aleksandr Livievich Samorodov Aleksandr Vladimirovich Bashirova Linara Irekovna Urakova Natalya Aleksandrovna Purygin Petr Petrovich Ermokhin Vladimir Anatolevich Bondareva Nataliya Aleksandrovna	RU2727508C1

RU 2 640 579 C1

Authors

Khaliullin Ferkat Adelzyanovich

Shabalina Yuliya Viktorovna

Samorodov Aleksandr Vladimirovich

Kamilov Feliks Khusainovich

Mustafin Ilshat Ganievich

Dates

2018-01-10—Published

2017-04-10—Filed