NEW N-ARYLSULPHAMIDE DERIVATIVE OF O-BENZOILAMINE-BENZOIC ACID WITH ANXIOLYTIC, ACTOPROTECTIVE AND ANTIDEPRESSANT ACTIVITY Russian patent published in 2018 - IPC C07D239/69 A61P25/24 A61P25/22 A61P37/02 

Abstract RU 2643356 C2

FIELD: pharmacology.

SUBSTANCE: invention relates to a new 2-benzoilamino-N-[4-(4,6-dimethylpyrimidine-2-ylsulfamoyl)-phenyl]-benzamide of the formula (I) having anxiolytic, actoprotective and antidepressant activity. The compound corresponds to the formula

, is low-toxic, and has a less pronounced effect on the leukocyte blood formula in chronic use, in contrast to diazepam.

EFFECT: compound can be used to obtain drugs for treatment of neuroses, neurotic states, psychopathies, affective, depressive, psychosomatic disorders, accompanied by emotional stress and anxiety disorders.

2 cl, 9 tbl, 1 ex

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RU 2 643 356 C2

Authors

Oganesyan Eduard Tonikovich

Kodonidi Ivan Panajotovich

Manvelyan Eleonora Aslibekovna

Sochnev Vadim Sergeevich

Sysa Valeriya Yurevna

Manvelyan Mikael Mikhajlovich

Dates

2018-02-01Published

2016-06-22Filed