DERIVATIVES OF 3-ALKYL-5-FLUORINE-4-SUBSTITUTED-IMINO-3,4-DIGIDROPYRIMIDINE-2 (H) -ONE AS FUNGICIDES Russian patent published in 2018 - IPC A01N43/54 A01P3/00 A61K31/513 

Abstract RU 2644014 C2

FIELD: chemistry.

SUBSTANCE: compound of the Formula I: , where R1 represents: C1-C6 alkyl, optionally substituted by 1-3 R4; -C(=O)R5; -C(=O)OR5; -CH2OC(=O)R5; or -(CHR8)nR7; R2 represents: C1-C6 alkyl, optionally substituted by 1-3 R6; -C(=O)R7; -C(=O)OR7; or -(CHR8)nR7, where n is an integer from 1-3; R3 represents -S(O)2R9; R4 independently represents C1-C6 alkyl, C1-C4 alkoxy, C1-C4 halogenoalkane, C1-C4 alkylthio, C1-C4 halogenalkyls, amino, C1-C3 alkylamino, C2-C6 alkoxycarbonyl, C2-C6 alkylsulphonyl, C2-C6 alkylaminocarbonyl, hydroxyl, deuterium, or C3-C6 trialkylsilyl; R5 represents N, C1-C6 alkyl, C2-C6 of alkenyl, C3-C6 alkynyl, C1-C6 halogenalkyls, C1-C6 alkoxyalkyl, phenyl or benzyl, where each of the phenyl or the benzyl may be optionally substituted by 1-3 R10, or a 5- or 6-membered saturated or unsaturated ring system, or 5 or 6 of the condensed ring system, or 6-6 condensed ring system each containing 1-3 heteroatom, where each ring may be optionally substituted by 1-3 R10, naftilan or biphenyl optionally substituted by 1-3 R10; R6 represent independently halogen, C1-C6 alkyl, C1-C4 halogenalkyls, C1-C4 alkoxy, C1-C4 halogenoalkane, C1-C4 alkylthio, C1-C4 halogenalkyls, amino, C1-C3 alkylamino, C2-C6 alkoxycarbonyl, C2-C6 alkylsulphonyl, C2-C6 alkylaminocarbonyl, hydroxyl, deuterium, or C3-C6 trialkylsilyl; R7 represents N, C1-C6 alkyl, C2-C6 of alkenyl, C3-C6 alkynyl, C1-C6 halogenalkyls, C1-C6 alkoxyalkyl, phenyl or benzyl, where each of the phenyl or the benzyl may be optionally substituted by 1-3 R10, or a 5- or 6-membered saturated or unsaturated ring system, or 5 or 6 of the condensed ring system, or 6-6 condensed ring system each containing 1-3 heteroatom, where each ring may be optionally substituted by 1-3 R10, naftilan or biphenyl optionally substituted by 1-3 R10; R8 represents N, C1-C6 alkyl or C1-C6 halogenalkyls; R9 represents1-C6 alkyl, C1-C6 halogenalkyls, amino, C1-C6 alkylamino, C2-C6 dialkylamino, phenyl or benzyl, where each of the phenyl or the benzyl may be optionally substituted by 1-3 R10, or 5- or 6-membered saturated or unsaturated ring containing 1-3 heteroatom, where each ring may be optionally substituted by 1-3 R10 or 5 or 6 of the condensed ring system, or 6-6 condensed ring system each containing 1-3 heteroatom, where each ring may be optionally substituted by 1-3 R10, naftilan or biphenyl optionally substituted by 1-3 R10; and R10 represent independently halogen, C1-C6 alkyl, C1-C4 halogenalkyls, C1-C4 alkoxy, C1-C4 halogenoalkane, C1-C4 alkylthio, C1-C4 halogenalkyls, amino, C1-C6 alkylamino, C2-C6 alkoxycarbonyl, C2-C6 alkylsulphonyl, C2-C6 alkylaminocarbonyl, C2-C6 dialkylamino, hydroxy, cyano or nitro.

EFFECT: invention makes it possible to increase the effectiveness of the control of phytopathogens.

21 cl, 3 tbl, 16 ex

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RU 2 644 014 C2

Authors

Lorsbakh Bet

Ross Ronald

Ouen U. Dzhon

Vebster Dzheffri D.

Stelzer Lindsej

Yao Chenlin

Lepla Pol

Gelliford Kristofer

Dates

2018-02-07Published

2013-12-23Filed