BIVALENT INHIBITORS OF IAP PROTEINS AND THERAPEUTIC METHODS OF IMPLEMENTATION Russian patent published in 2018 - IPC C07D487/04 C07D519/00 A61K31/395 A61P35/00 

Abstract RU 2649975 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention relates to structure compounds

, as well as to their pharmaceutically acceptable salts.

EFFECT: technical result: new compounds are obtained that are inhibitors of IAP proteins, as well as pharmaceutical compositions based on them, suitable for treatment of diseases and conditions, in which inhibition of IAP protein provides a benefit, like cancers.

14 cl, 1 dwg, 50 ex, 1 tbl

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RU 2 649 975 C2

Authors

Van Shaomen

Shen Zhun

Sun Khajin

Lyu Lyu

Lu Tszyanfen

Makichern Donna

Dates

2018-04-06Published

2013-08-16Filed