5-ETHYL-2-AMINO-1,3,4-THIADIAZOLE DERIVATIVES WITH ANESTHETIC, ANTI-INFLAMMATORY, ANTI-ALLERGIC AND ANALGETIC ACTIVITY Russian patent published in 2018 - IPC C07D285/135 A61K31/433 A61P29/00 

Abstract RU 2651572 C2

FIELD: pharmacology.

SUBSTANCE: invention relates to 5-ethyl-2-amino-1,3,4-thiadiazole derivatives, namely N-(5-ethyl-1,3,4-thiadiazol-2-yl)-amide of N-acetylaminohexanoic acid

(compound 1 ),

5-ethyl-2-amino-1,3,4-thiadiazole succinate

(compound 2 ),

5-ethyl-2-amino-1,3,4-thiadiazole D,L-hydroxysuccinate

(compound 3 ).

EFFECT: 5-ethyl-2-amino-1,3,4-thiadiazole derivatives have anesthetic, anti-inflammatory, anti-allergic and analgesic activities.

6 tbl, 4 ex

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RU 2 651 572 C2

Authors

Skachilova Sofiya Yakovlevna

Zheltukhin Nikolaj Konstantinovich

Demidova Marina Aleksandrovna

Popov Nikita Sergeevich

Kazaishvili Yurij Georgievich

Korotonozhkin Aleksej Viktorovich

Proskurina Oksana Vladimirovna

Olkhovich Marina Vasilevna

Perlovich German Leonidovich

Dates

2018-04-23Published

2016-08-05Filed