N-(5-ETHYL-1,3,4-TIADIAZOL-2-YL)-2-PROPYLPENTANAMID, POSSESSING ANTIEPILEPTIC AND ANALGESIC ACTIVITIES Russian patent published in 2018 - IPC C07D285/135 A61K31/433 A61P25/08 A61P29/00 

Abstract RU 2672887 C1

FIELD: chemistry.

SUBSTANCE: present invention relates to a new biologically active compound, in particular to N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-propylpentanamide of the following formula:

,

that has antiepileptic and analgesic activities.

EFFECT: obtaining a new derivative of 1,3,4-thiadiazole with 2-propylpentanoic acid, characterized by low toxicity, suggesting its effective use in medicine as a means to treat neuropathic pain and epilepsy.

1 cl, 4 tbl, 5 ex

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RU 2 672 887 C1

Authors

Skachilova Sofiya Yakovlevna

Malygin Aleksandr Sergeevich

Popov Nikita Sergeevich

Demidova Marina Aleksandrovna

Sadchikova Natalya Petrovna

Zheltukhin Nikolaj Konstantinovich

Korotonozhkin Aleksej Viktorovich

Dates

2018-11-20Published

2018-03-13Filed