FIELD: medicine.
SUBSTANCE: invention relates to medicine, namely to pharmaceutical composition for modulating the activity of glutaminyl cyclase, and also for treatment of a disorder associated with glutaminyl cyclase activity containing an effective amount of a compound of N,N'-bis[2-(1H-imidazol-4-yl)ethyl]isophthalamide.
.
EFFECT: implementation of invention will yield effective glutaminyl cyclase modulator having a high activity with respect to intracellular and/or secreted isoforms of glutaminyl cyclase and good pharmacokinetic characteristics.
11 cl, 10 ex, 6 tbl
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