NEW GLUTAMINE CYCLASE INHIBITOR AND ITS APPLICATION Russian patent published in 2023 - IPC C07D403/12 A61K31/4174 A61P1/02 A61P13/12 A61P43/00 

Abstract RU 2791703 C2

FIELD: medicine.

SUBSTANCE: suggested is the use of N,N'-bis[2-(1H-imidazol-4-yl)ethyl]isophthalamide or its pharmaceutically acceptable salt, hydrate or solvate for the treatment of a disorder, Crohn's disease, ulcerative colitis, peritonitis, nephropathy, or kidney disease, which is a side effect of the use of drugs. Also provided is a process for treating the disease, including administration of the said compound in a therapeutically effective amount.

EFFECT: technical result is the use of a compound that is effective in modulating glutaminyl cyclase in the treatment of diseases associated with aberrant activity of immune system cells.

4 cl, 6 tbl, 9 ex

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RU 2 791 703 C2

Authors

Nebolsin Vladimir Evgenevich

Kromova Tatyana Aleksandrovna

Rydlovskaya Anastasiya Vladimirovna

Dates

2023-03-13Published

2018-08-09Filed