PIPERIDINE UREA DERIVATIVES Russian patent published in 2018 - IPC C07D401/14 C07D401/06 C07D401/12 C07D401/08 C07D211/46 A61K31/445 A61K31/4545 A61P35/00 A61P25/28 

Abstract RU 2666894 C2

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to piperidine urea derivatives, Claim 1, and to their pharmaceutically acceptable salts. Invention also relates to drugs which inhibit the activity of Tankyrases (TANKs) and poly(ADP-ribose)polymerase PARP-1, based on these compounds.

EFFECT: new compounds have been obtained that can be used in medicine for the treatment of diseases such as malignant neoplasm, cardiovascular diseases, central nervous system lesions and various forms of inflammation.

2 cl, 3 tbl, 37 ex

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RU 2 666 894 C2

Authors

Bukhshtaller Khans-Peter

Dorsh Diter

Dates

2018-09-13Published

2014-07-09Filed