FIELD: pharmaceuticals.
SUBSTANCE: invention relates to piperidine urea derivatives, Claim 1, and to their pharmaceutically acceptable salts. Invention also relates to drugs which inhibit the activity of Tankyrases (TANKs) and poly(ADP-ribose)polymerase PARP-1, based on these compounds.
EFFECT: new compounds have been obtained that can be used in medicine for the treatment of diseases such as malignant neoplasm, cardiovascular diseases, central nervous system lesions and various forms of inflammation.
2 cl, 3 tbl, 37 ex
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Authors
Dates
2018-09-13—Published
2014-07-09—Filed