MULTISUBSTITUTED AROMATIC COMPOUNDS AS SERINE PROTEASE INHIBITORS Russian patent published in 2019 - IPC A61K31/4439 A61P43/00 

Abstract RU 2678830 C2

FIELD: medicine.

SUBSTANCE: group of inventions relates to medicine, namely to pharmaceutical industry. Compound having the structure of formula (V):

as well as a pharmaceutical composition containing a therapeutically effective amount of compound (V) are proposed.

EFFECT: use of the inventions provides a wider range of agents exhibiting inhibitory action against serine proteases - thrombin and kallikrein.

25 cl, 5 tbl, 37 ex

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RU 2 678 830 C2

Authors

Short Kevin Majkl

Fam Son Minkh

Uillyams Devid Charlz

Kita Devid Ben

Dates

2019-02-04Published

2014-03-17Filed