MULTI-SUBSTITUTED AROMATIC COMPOUNDS AS THROMBIN INHIBITORS Russian patent published in 2017 - IPC C07D401/04 C07D405/14 C07D409/14 A61K31/4439 A61K31/4427 A61P7/02 A61P7/00 A61P25/28 

Abstract RU 2639876 C2

FIELD: pharmacology.

SUBSTANCE: invention relates to a compound of the formula: , and also to pharmaceutical compositions and methods for treatment and prevention of a disease such as thrombotic one.

EFFECT: new compounds capable of inhibiting the protease activity of thrombin.

15 cl, 3 tbl, 85 ex

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RU 2 639 876 C2

Authors

Short Kevin Majkl

Fam Son Minkh

Uillyams Devid Charlz

Datta Somalee

Dates

2017-12-25Published

2011-03-30Filed