Show metadata Hide metadata

(19)

(11)

2 686 323

(13)

(51)

IPC

C07D295/192(2006-01-01)

A61K31/4965(2006-01-01)

A61K35/00(2006-01-01)

(21) (22)

Application

2015141772, 2014-03-11

(24)

Start date

2014-03-11

(22)

Actual filing date

2014-03-11

(45)

Published

2019-04-25

(72)

Inventor

Bejr Kennet V.Lancha Devid R.Li KhunbinLok DzhejmsLyu VejMartin Mettyu V.Millan Devid S.Shiller Shon E.R.Tebbe Mark Dzh.

(73)

Holder

Forma Terapyutiks, Ink.

NOVEL COMPOUNDS AND COMPOSITIONS FOR INHIBITION OF FASN Russian patent published in 2019 - IPC C07D295/192 A61K31/4965 A61K35/00

Abstract RU 2686323 C2

FIELD: chemistry.

SUBSTANCE: invention relates to compounds of formula I-B, as well as to pharmaceutical compositions based on them.

EFFECT: obtained are novel compounds with the ability to inhibit fatty acid synthase (FASN).

31 cl, 6 tbl

Similar patents RU2686323C2

Title	Year	Author	Number
NOVEL COMPOUNDS AND FASN INHIBITION COMPOSITIONS	2014	Bair, Kenneth, W. Lancia, David, R. Li, Hongbin Loch, James Lu, Wei Martin, Matthew, W. Millan, David, S. Schiller, Shawn, E.R. Tebbe, Mark, J.	RU2737434C2
BICYCLIC COMPOUNDS AS PD1/PD-L1 INTERACTION/ACTIVATION INHIBITORS	2019	Venkateshappa, Chandregowda D A, Jeyaraj Pendyala, Muralidhar Sivanandhan, Dhanalakshmi Rajagopal, Sridharan	RU2777980C2
MONOMER DERIVATIVES OF GLYCOPEPTIDE ANTIBIOTIC	2005	Arimoto Khirokazu Lu Tszjun' Jamano Josinori Jasukata Tatsuro Josida Osamu Ivaki Tsutomu Josida Jutaka Kato Issei Morimoto Kendzi Jasosima Kajo	RU2424248C2
THERAPEUTICALLY ACTIVE DERIVATIVES OF OXAZOLINE	2013	Kulisa Kler Luiz Brukings Deniel Kristofer Ford Deniel Dzhejms Franklin Richard Dzheremi Rojberson Dzhejms Tomas Gavalkar Anant Ramrao	RU2656209C2
PYRAZOLOPYRIDINE DERIVATIVES AS KINASE INHIBITORS	2015	Ford Daniel Dzhejms Ryuberson Dzhejms Tomas	RU2733400C2
NOVEL COMPOUNDS AND COMPOSITIONS FOR INHIBITING NAMPT	2011	Bejr Kennet V. Baumajster Timm R. Bakmelter Aleksandr Dzh. Klodfelter Karl Kh. Khan Binsun Lin Tszyan Rejnolds Dominik Dzh. Smit Chejz K. Van Chzhungo Chzhen Syaochzhan Yuen Po-Vaj	RU2617424C2
HETEROCYCLIC COMPOUNDS AND USES THEREOF	2014	Chzhan Tszyayazhun Buell Dzhon Chan Katrina Ibrakhim Prabkha N. Lin Dzhek Fam Fuongli Shi Sonyuan Spevak Vejn Vu Guosyan Vu Dzheffri	RU2680100C9
METHOD FOR PRODUCTION OF HYDROXYLATED CYCLOPENTYL PYRIMIDINE COMPOUNDS	2013	Askin Devid Khan Chun Lejn Dzhonatan V. Remarchuk Trevis Shakya Sagar Sauell K. Gregori Spenser Kejt L. Stendzhel Piter Dzh.	RU2643811C2
DIHYDROPYRIDAZINE-3,5-DIONE DERIVATIVE	2014	Okhtake Josikhito Okamoto Naoki Ono Esiyuki Kasivagi Khirotaka Kimbara Atsusi Kharada Takeo Khori Nobuyuki Murata Esikhisa Tatibana Kadzutaka Tanaka Sota Nomura Keniti Ide Mitsuaki Midzuguti Ejsaku Itida Yasukhiro Okhtomo Suiti Khoriba Naosi	RU2662832C2
INDOL-3-YL-CARBONYL-ASASPIRO DERIVATIVES AS VASOPRESSIN RECEPTOR ANTAGONISTS	2006	Bissants Katerina Grundshober Kristof Ratni Khasan Rodzhers-Ehvans Mark Shnajder Patrik	RU2418801C2

RU 2 686 323 C2

Authors

Bejr Kennet V.

Lancha Devid R.

Li Khunbin

Lok Dzhejms

Lyu Vej

Martin Mettyu V.

Millan Devid S.

Shiller Shon E.R.

Tebbe Mark Dzh.

Dates

2019-04-25—Published

2014-03-11—Filed