NOVEL COMPOUNDS AND COMPOSITIONS FOR INHIBITING NAMPT Russian patent published in 2017 - IPC C07D213/54 C07D213/38 C07D213/74 C07D471/04 C07C317/14 A61K31/4406 A61P35/00 

Abstract RU 2617424 C2

FIELD: chemistry.

SUBSTANCE: invention relates to compounds of formula IIIA

.

EFFECT: obtaining novel compounds of formula IIIA, as well as compositions based thereon for inhibiting NAMPT, described is use of compounds for preparing a drug for treating cancer.

21 cl, 3 tbl, 20 ex, 3 dwg

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RU 2 617 424 C2

Authors

Bejr Kennet V.

Baumajster Timm R.

Bakmelter Aleksandr Dzh.

Klodfelter Karl Kh.

Khan Binsun

Lin Tszyan

Rejnolds Dominik Dzh.

Smit Chejz K.

Van Chzhungo

Chzhen Syaochzhan

Yuen Po-Vaj

Dates

2017-04-25Published

2011-09-02Filed