HALOGEN SUBSTITUTED HETEROCYCLIC COMPOUND SALT Russian patent published in 2019 - IPC C07D333/36 A61K31/381 A61P1/16 A61P11/00 A61P13/12 

Abstract RU 2689315 C2

FIELD: chemistry.

SUBSTANCE: invention relates to salts of a thiophene compound substituted with α-halogen of general formula (I):

(I), (where R denotes a hydrogen atom or a methoxy group; X is a halogen atom; A is selected from a group consisting of; M is an alkali or alkali-earth metal; and n is 1 when M is an alkali metal, and is 2 when M is an alkali-earth metal).

EFFECT: compound possesses strong LPA receptor antagonist action.

15 cl, 1 tbl, 45 ex

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RU 2 689 315 C2

Authors

Iwase, Noriaki

Nishida, Hiroshi

Okudo, Makoto

Ito, Masaaki

Kono, Shigeyuki

Matoyama, Masaaki

Ushiyama, Shigeru

Okanari, Eiji

Matsunaga, Hirofumi

Nishikawa, Kenji

Kimura, Tomio

Dates

2019-05-27Published

2015-06-26Filed