PIPERAZINE DERIVATIVES, CHARACTERIZED BY MULTIMODAL ACTIVITY ON PAIN Russian patent published in 2019 - IPC C07D231/12 C07D249/04 C07D249/14 C07D401/14 C07D403/06 A61K31/496 A61P25/00 

Abstract RU 2709482 C1

FIELD: medicine; pharmaceuticals; chemistry.

SUBSTANCE: invention refers to compounds of formula (I), methods for preparing them and pharmaceutical compositions containing them.

EFFECT: technical result: obtaining novel compounds having double pharmacological activity with respect to sigma (σ1) receptor, and μ-opioid receptor, which can be used for treatment, in particular for pain management.

13 cl, 2 tbl, 2 ex

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RU 2 709 482 C1

Authors

Kuevas Kordobes Feliks

Almansa-Rosales Karmen

Garsiya Lopes Monika

Dates

2019-12-18Published

2014-12-19Filed