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(19)

RU

(11)

2 712 272

(13)

C2

(51)

IPC

C07D417/14(2006-01-01)

A61K31/541(2006-01-01)

A61P25/28(2006-01-01)

(21) (22)

Application

2017134884, 2016-03-16

(24)

Start date

2016-03-16

(22)

Actual filing date

2016-03-16

(45)

Published

2020-01-28

(72)

Inventor

Bartels BernDolente KozimoGuba VolfgangKhaap VolfgangObst Zander UlrikePeters Jens-UveVoltering Tomas

(73)

Holder

F. Hoffmann-La Roche Ag

BETA-SECRETASE INHIBITORS Russian patent published in 2020 - IPC C07D417/14 A61K31/541 A61P25/28 

Abstract RU 2712272 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention refers to compounds of formula I, as well as to pharmaceutical compositions based thereon.

EFFECT: technical result is obtaining novel compounds having BACE1 inhibitor activity, useful in therapeutic and/or preventive treatment of mediated diseases.

22 cl, 9 tbl, 44 ex

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RU 2 712 272 C2

Authors

Bartels Bern

Dolente Kozimo

Guba Volfgang

Khaap Volfgang

Obst Zander Ulrike

Peters Jens-Uve

Voltering Tomas

Dates

2020-01-28—Published

2016-03-16—Filed

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