PYRIDAZINONE DERIVATIVES AS PARP INHIBITORS Russian patent published in 2013 - IPC C07D403/10 C07D403/12 A61K31/501 A61P29/00 

Abstract RU 2490265 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to compounds of formula (I): . Therein the values A, R1, R2, R6, r, Rc are presented in cl.1 of the patent claim, as well as to pharmaceutically acceptable salts or tautomers of the above compound being poly(ADP-ribose)polymerase (PARP) inhibitors.

EFFECT: preparing the pharmaceutically acceptable salts or tautomers of the above compound being poly(ADP-ribose)polymerase (PARP) inhibitors.

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RU 2 490 265 C2

Authors

Branka Danila

Dessole Gabriehlla

Ferrin'O Federika

Dzhouns Filip

Kintsel' Olaf

Lillini Samuehle

Mural'Ja Ehster

Peskatore Dzhovanna

Shul'Tts-Fademrekht Karsten

Dates

2013-08-20Published

2008-11-14Filed