Patenton — panteon of patents

(19)

RU

(11)

2 720 237

(13)

C2

(51)

IPC

C07D241/42(2006-01-01)

A61K31/53(2006-01-01)

A61K31/4985(2006-01-01)

A61P3/04(2006-01-01)

A61P15/16(2006-01-01)

A61P19/02(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2016124178, 2014-11-18

(24)

Start date

2014-11-18

(22)

Actual filing date

2014-11-18

(45)

Published

2020-04-28

(72)

Inventor

Bair Kenneth W.Herbertz TorstenKauffman Goss StrykerKayser-Bricker Katherine J.Luke George P.Martin Matthew W.Millan David S.Schiller Shawn E. R.Talbot Adam C.Tebbe Mark J.

(73)

Holder

Forma Therapeutics, Inc.

COMPOSITIONS CONTAINING BENZOPIPERAZINE AS BROMODOMAIN BET INHIBITORS Russian patent published in 2020 - IPC C07D241/42 A61K31/53 A61K31/4985 A61P3/04 A61P15/16 A61P19/02 A61P35/00 

Abstract RU 2720237 C2

FIELD: pharmaceuticals.

SUBSTANCE: present invention relates to compounds of formula (VI), as well as to pharmaceutical compositions based thereon.

EFFECT: technical result is obtaining novel compounds exhibiting properties of bromodomain family (BET) inhibitors.

16 cl, 34 tbl, 288 ex

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RU 2 720 237 C2

Authors

Bair Kenneth W.

Herbertz Torsten

Kauffman Goss Stryker

Kayser-Bricker Katherine J.

Luke George P.

Martin Matthew W.

Millan David S.

Schiller Shawn E. R.

Talbot Adam C.

Tebbe Mark J.

Dates

2020-04-28—Published

2014-11-18—Filed

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