FIELD: medicine; pharmaceuticals.
SUBSTANCE: invention relates to a polymorph of bis-mesylate salt of 3-(3-(4-(1-aminocyclobutyl)phenyl)-5-phenyl-3H-imidazo[4,5-b]pyridin-2-yl)pyridin-2-amine (compounds A), forms A, B, C, D, E and I. Invention also relates to a pharmaceutical composition on a polymorph of compound A and a method of treating or preventing a cell proliferation disorder in a subject in need thereof.
(A).
EFFECT: polymorph of bis-mesylate salt of 3-(3-(4-(1-aminocyclobutyl)phenyl)-5-phenyl-3H-imidazo[4,5-b]pyridin-2-yl)pyridin-2-amine, having useful biological properties.
33 cl, 21 tbl, 40 ex, 263 dwg
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