CONJUGATE SALTS FOR CANCER TREATMENT Russian patent published in 2021 - IPC C07H19/06 A61K47/50 A61P35/00 A61P35/02 

Abstract RU 2747528 C2

FIELD: biochemistry.

SUBSTANCE: invention relates to pharmacologically acceptable salts, represented by the structure of Formula (1), which can be used for the treatment of cancer or a precancerous condition or disorder. In Formula (1), Y is a pharmacologically acceptable organic or inorganic acid or acid residue, with the specified acid selected from HCl, methanesulfonic acid, trifluoroacetic acid (TFA), H2SO4 and H3PO4. The invention also relates to a pharmaceutical composition containing these salts and methods for the treatment of cancer or a precancerous condition, including in a subject who has an immunological disease or a disorder or dysfunction of organs.

EFFECT: invention may find application treatment of cancer or a precancerous condition or disorder.

22 cl, 5 dwg, 5 tbl, 24 ex

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RU 2 747 528 C2

Authors

Gengrinovich, Stela

Dates

2021-05-06Published

2016-12-01Filed