Show metadata Hide metadata

(19)

(11)

2 748 748

(13)

(51)

IPC

C07D265/36(2006-01-01)

A61K31/538(2006-01-01)

A61P31/06(2006-01-01)

(21) (22)

Application

2020121634, 2020-06-25

(24)

Start date

2020-06-25

(22)

Actual filing date

2020-06-25

(45)

Published

2021-05-31

(72)

Inventor

Maslivets Andrej NikolaevichMashevskaya Irina VladimirovnaBalandina Svetlana YurevnaStepanova Ekaterina EvgenevnaDmitriev Maksim ViktorovichKovalenko Ilya IvanovichDrobkova Vera AnatolevnaRemezovskaya Natalya Borisovna

(73)

Holder

Federalnoe Gosudarstvennoe Avtonomnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniya Gosudarstvennyj Natsionalnyj Issledovatelskij Universitet"

ANTI-TUBERCULOSIS DRUG BASED ON (Z)-3-(3,3-DIMETHYL-2-OXOBUTYLIDENE) -3,4-DIHYDRO-2H-1,4-BENZOXAZIN-2-ONE AND A METHOD FOR ITS SYNTHESIS Russian patent published in 2021 - IPC C07D265/36 A61K31/538 A61P31/06

Abstract RU 2748748 C1

FIELD: pharmaceutical industry.

SUBSTANCE: invention relates to (Z) -3- (3,3-dimethyl-2-oxobutylidene) -3,4-dihydro-2H-1,4-benzoxazin-2-one with anti-tuberculosis activity.

EFFECT: use of (Z) -3- (3,3-dimethyl-2-oxobutylidene) -3,4-dihydro-2H-1,4-benzoxazin-2-one as an anti-tuberculosis agent is proposed.

1 cl, 4 ex, 5 tbl

Similar patents RU2748748C1

Title	Year	Author	Number
DIALKYL(2-METHYL-4-OXOPENT-2-YL)PHOSPHINE OXIDE PYRIDINOYL HYDRAZONES, HAVING ANTITUBERCULOUS ACTIVITY	2012	Kostin Anton Alekseevich Tatarinov Dmitrij Anatol'Evich Kashapov Lenar Ramilovich Chestnova Regina Valer'Evna Valiev Ravil' Shamilovich Garaev Ramil Sufiakhmetovich Buzykin Boris Ivanovich Mironov Vladimir Fedorovich	RU2498990C1
DIMEPHOSPHONE ISONICOTINOYLHYDRAZONE WITH ANTI-TUBERCULOSIS ACTIVITY	2011	Buzykin Boris Ivanovich Nabiullin Vazikh Nurulaevich Mironov Vladimir Fedorovich Chestnova Regina Valer'Evna Garaev Ramil Sufiakhmetovich Kashapov Lenar Ramilovich Mironova Ekaterina Vladimirovna Tatarinov Dmitrij Anatol'Evich Kostin Anton Alekseevich	RU2457212C1
DIMEPHOSPHONE NICOTINOYLHYDRAZONE POSSESSING ANTI-TUBERCULOSIS ACTIVITY	2011	Buzykin Boris Ivanovich Nabiullin Vazikh Nurulaevich Mironov Vladimir Fedorovich Chestnova Regina Valer'Evna Garaev Ramil Sufiakhmetovich Kashapov Lenar Ramilovich Mironova Ekaterina Vladimirovna Tatarinov Dmitrij Anatol'Evich Kostin Anton Alekseevich	RU2471787C1
COMBINED ANTITUBERCULOUS COMPOSITION	2009	Mokhireva Ljudmila Vikent'Evna Erokhin Vladislav Vsevolodovich Robakidze Tat'Jana Nikolaevna Emshanova Svetlana Vital'Evna Mokhirev Aleksej Vladimirovich	RU2413517C1
ANTI-TUBERCULOSIS AGENT BASED ON 4-((HET)AROYL)-3-HYDROXY-1-(2-HYDROXYPHENYL)-5-(PHENYLTHIO)-1,5-DIHYDRO-2H-PYRROL-2-ONES	2021	Mashevskaya Irina Vladimirovna Balandina Svetlana Yurevna Lukmanova Dzhamilya Nailevna	RU2767542C1
5-FLUORO-2-(4-ETHOXYCARBONYLDIPIPERAZINE-1-YL)-1,3-BENZOTHIAZINE-4-ONE, WHICH HAS ANTI-TUBERCULOSIS ACTIVITY	2018	Charushin Valerij Nikolaevich Nosova Emiliya Vladimirovna Poteeva Anna Dmitrievna Kotovskaya Svetlana Konstantinovna Lipunova Galina Nikolaevna Kravchenko Marionella Anatolevna Skornyakov Sergej Nikolaevich Medvinskij Igor Davydovich	RU2663848C1
TRAIZINES HAVING ANTI-TUBERCULOSIS ACTIVITY	2010	Fattakhov Saitgarej Galjauvich Valiev Ravil' Shamilovich Shulaeva Marina Mikhajlovna Sajfina Lilija Fuadovna Chestnova Regina Valer'Evna Mingaleev Danil Nail'Evich Tremasov Mikhail Jakovlevich Ravilov Rustam Khametovich Reznik Vladimir Savich	RU2431633C1
COMBINED ANTITUBERCULOUS COMPOSITION	2010	Mokhireva Ljudmila Vikent'Evna Emshanova Svetlana Vital'Evna Mokhirev Aleksej Vladimirovich	RU2468802C2
METHOD OF TREATING TUBERCULOSIS WITH MULTIPLE DRUG RESISTANCE	2013	Sharma Radzhesh Vasil'Eva Irina Anatol'Evna	RU2554753C2
SALT OF BIS(OXYMETHYL)PHOSPHINIC ACID WITH ISONICOTINIC ACID HYSRAZIDE (TUBOPHEN) HAVING ANTITUBERCULOSIS ACTION AND METHOD FOR PRODUCTION THEREOF	2005	Fattakhov Saitgarej Galjauvich Mingaleev Danil Nail'Evich Safin Marat Abdrakhmanovich Reznik Vladimir Savich Zaljalov Il'Dar Nadyrovich Tremasov Mikhail Jakovlevich Konovalov Aleksandr Ivanovich Vizel' Aleksandr Andreevich	RU2281939C1

RU 2 748 748 C1

Authors

Maslivets Andrej Nikolaevich

Mashevskaya Irina Vladimirovna

Balandina Svetlana Yurevna

Stepanova Ekaterina Evgenevna

Dmitriev Maksim Viktorovich

Kovalenko Ilya Ivanovich

Drobkova Vera Anatolevna

Remezovskaya Natalya Borisovna

Dates

2021-05-31—Published

2020-06-25—Filed