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2 663 848

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IPC

C07D417/04(2006-01-01)

A61K31/5415(2006-01-01)

A61P31/06(2006-01-01)

(21) (22)

Application

2018110471, 2018-03-23

(24)

Start date

2018-03-23

(22)

Actual filing date

2018-03-23

(45)

Published

2018-08-10

(72)

Inventor

Charushin Valerij NikolaevichNosova Emiliya VladimirovnaPoteeva Anna DmitrievnaKotovskaya Svetlana KonstantinovnaLipunova Galina NikolaevnaKravchenko Marionella AnatolevnaSkornyakov Sergej NikolaevichMedvinskij Igor Davydovich

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Uchrezhdenie Nauki Institut Organicheskogo Sinteza Im. I.Ya. Postovskogo Uralskogo Otdeleniya Rossijskoj Akademii Nauk Uro Ran)Federalnoe Gosudarstvennoe Byudzhetnoe Uchrezhdenie Meditsinskij Issledovatelskij Tsentr Ftiziopulmonologii I Infektsionnykh Zabolevanij" Ministerstva Zdravookhraneniya Rossijskoj Federatsii Fpi" Minzdrava Rossii)

5-FLUORO-2-(4-ETHOXYCARBONYLDIPIPERAZINE-1-YL)-1,3-BENZOTHIAZINE-4-ONE, WHICH HAS ANTI-TUBERCULOSIS ACTIVITY Russian patent published in 2018 - IPC C07D417/04 A61K31/5415 A61P31/06

Abstract RU 2663848 C1

FIELD: chemistry.

SUBSTANCE: invention relates to the field of organic chemistry, namely 5-fluoro-2-(4-ethoxycarbonylpiperazine-1-yl)-1,3-benzothiazine-4-one of formula (4) having anti-tuberculosis activity, including in relation to strains of mycobacteria with multiple drug resistance. 4.

EFFECT: new heterocyclic compound having useful biological properties has been obtained.

1 cl, 4 tbl, 1 ex

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RU 2 663 848 C1

Authors

Charushin Valerij Nikolaevich

Nosova Emiliya Vladimirovna

Poteeva Anna Dmitrievna

Kotovskaya Svetlana Konstantinovna

Lipunova Galina Nikolaevna

Kravchenko Marionella Anatolevna

Skornyakov Sergej Nikolaevich

Medvinskij Igor Davydovich

Dates

2018-08-10—Published

2018-03-23—Filed