CRYSTALLINE FORM OF THE COMPOUND CONSTITUTING A PRODRUG OF LANOSTEROL, AND APPLICATION THEREOF IN MANUFACTURE OF A MEDICINAL PRODUCT FOR TREATING CATARACTS Russian patent published in 2022 - IPC C07J9/00 A61K9/08 A61K31/573 A61P27/12 

Abstract RU 2766088 C1

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to the crystalline form A of the compound by the formula (I), wherein the X-ray powder diffractogram (XPRD) of the crystalline form A comprises characteristic diffraction peaks at the following values of the angle 2θ: 8.60±0.2°, 9.38±0.2°, 10.57±0.2°, 12.54±0.2°, 14.43±0.2°, 15.06±0.2°, 17.22±0.2°, and 25.18±0.2°. The crystalline form of the compound by the formula (I) is intended for application for producing a medicinal product for treating cataracts.

EFFECT: crystalline form A of the compound by the formula (I), exhibiting good stability.

8 cl, 10 dwg, 6 tbl, 3 ex

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RU 2 766 088 C1

Authors

Liu, Yizhi

Wang, Yandong

Li, Xiaolin

Luo, Zhi

He, Haiying

Li, Jian

Chen, Shuhui

Dates

2022-02-07Published

2019-07-25Filed