SUBSTITUTED THIOPHENECARBOXAMIDES AND ANALOGUES AS ANTIBACTERIAL AGENTS Russian patent published in 2023 - IPC C07D333/38 C07D333/40 C07D413/04 A01N43/10 A01N43/28 A01P1/00 

Abstract RU 2797316 C2

FIELD: organic chemistry.

SUBSTANCE: invention relates to a substituted thiophenecarboxamide of formula (I), where R1 and R2 are identical and represent a chlorine atom or a bromine atom; R3 is methyl; R4 is selected from the group consisting of a hydrogen atom, alkyl with 1–6 carbon atoms, benzyl atoms, and benzyl substituted with hydroxyl atoms, alkyl with 1–6 carbon atoms substituted with C1-C6-alkylsulfanyl, and R5 represents a hydrogen atom; or R4 and R5 together with the carbon atom to which they are attached form cyclopropyl; R6 is selected from the group consisting of hydrogen, alkyl with 1–6 hydrogen atoms, haloalkyl with 1–6 hydrogen atoms, cyanoalkyl with 3–8 hydrogen atoms, phenyl, benzyl, oxetanyl, -C1-C6-alkyl-Si(C1-C6-alkyl)3 and -C1-C6-alkyl-C3-C8-cycloalkyl. The invention also relates to intermediate compounds, the structures and meanings of which are indicated in the formula.

EFFECT: protection of plants from bacterial diseases, in particular, those caused by bacteria belonging to Xanthomonas genus.

8 cl, 8 tbl, 9 ex

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RU 2 797 316 C2

Authors

Bernier, David

Brunet, Stephane

Dufour, Jeremy

Knobloch, Thomas

Nicolas, Lionel

Tsuchiya, Tomoki

Dates

2023-06-02Published

2019-07-03Filed