N-(5-BROMOPYRIDIN-2-YL)-4-OXO-4-(P-TOLYL)-2-((3-CYANO-4,5,6,7-TETRAHYDROBENZO[B]THIOPHEN-2-YL) )AMINO)BUT-2-ENAMIDE AS AN ANTI-INFLAMMATORY DRUG Russian patent published in 2023 - IPC C07D409/12 A61K31/4436 A61P29/00 

Abstract RU 2798426 C1

FIELD: organic chemistry.

SUBSTANCE: invention relates to the field of organic chemistry, namely the use of N-(5-bromopyridin-2-yl)-4-oxo-4-(p-tolyl)-2-((3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)amino)but-2-enamide of formula 1 as a drug having anti-inflammatory activity.

EFFECT: N-(5-bromopyridin-2-yl)-4-oxo-4-(p-tolyl)-2-((3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl) amino)but-2-enamide, which has anti-inflammatory activity and low toxicity.

1 cl, 2 tbl, 3 ex

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RU 2 798 426 C1

Authors

Shipilovskikh Sergei Aleksandrovich

Makhmudov Ramiz Ragibovich

Gorbunova Irina Aleksandrovna

Okoneshnikova Elizaveta Aleksandrovna

Dates

2023-06-22Published

2022-07-01Filed