ANTIBODY-DRUG CONJUGATES AND THEIR USE FOR THE TREATMENT OF CANCER DISEASES Russian patent published in 2023 - IPC A61K47/65 A61K47/68 A61P35/00 

Abstract RU 2799547 C2

FIELD: medicine.

SUBSTANCE: invention relates to antibody-drug conjugates wherein the antibodies specifically bind to the transferrin receptor TFR and the drugs are preferably selected from cytotoxic agents. The invention relates to antibody-drug conjugates, where the antibodies specifically bind to the transferrin receptor TFR and the drug is monomethylauristatin E.

EFFECT: such antibody-drug conjugates can be used in particular in the treatment of proliferative diseases, including cancer diseases such as lymphomas or leukemias.

10 cl, 10 dwg, 8 tbl, 10 ex

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RU 2 799 547 C2

Authors

Launay, Pierre

Souchet, Herve

Belanger, Coralie

Dates

2023-07-06Published

2019-04-09Filed