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2 805 915

(13)

(51)

IPC

C07D493/04(2006-01-01)

C07D519/00(2006-01-01)

A61K31/34(2006-01-01)

A61K31/422(2006-01-01)

A61K31/506(2006-01-01)

A61K31/662(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2023104161, 2023-02-22

(24)

Start date

2023-02-22

(22)

Actual filing date

2023-02-22

(45)

Published

2023-10-24

(72)

Inventor

Salin Aleksei ValerevichVoloshina Aleksandra DmitrievnaAmerkhanova Siumbelia KamilevnaLiubina Anna Pavlovna

(73)

Holder

Federalnoe Gosudarstvennoe Avtonomnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniia Federalnyi Universitet» Vo Kfu)

ARGLABIN DERIVATIVES WITH SELECTIVE CYTOTOXIC EFFECTS Russian patent published in 2023 - IPC C07D493/04 C07D519/00 A61K31/34 A61K31/422 A61K31/506 A61K31/662 A61P35/00

Abstract RU 2805915 C1

FIELD: organic and medicinal chemistry.

SUBSTANCE: invention relates to the arglabin derivatives of formulas Ib, Ic, Id, Ie. New compounds that can be used in medicine as targeted antitumor medicinal products with low cytotoxicity towards normal cell lines have been obtained.

EFFECT: obtaining arglabin derivatives with selective cytotoxic effects.

4 cl, 2 dwg, 7 ex

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RU 2 805 915 C1

Authors

Salin Aleksei Valerevich

Voloshina Aleksandra Dmitrievna

Amerkhanova Siumbelia Kamilevna

Liubina Anna Pavlovna

Dates

2023-10-24—Published

2023-02-22—Filed