(2S)-3-(4-{2-[4-(2-{[(1R,4AR,7S)-7-ETHYNYL-1,4A,7-TRIMETHYL-1,2,3,4,4A,4B,5,6,7,8,10,10A-DODECAHYDROPHENANTHREN-1-YL]FORMAMIDO}ETHOXY)PHENYL]ETHOXY}PHENYL)-2-ETHOXY-PROPANOIC ACID FOR THERAPY AND PREVENTION OF METABOLIC SYNDROME Russian patent published in 2024 - IPC C07C43/205 C07J53/00 C07J63/00 A61P3/10 

Abstract RU 2813464 C1

FIELD: chemistry; pharmacology.

SUBSTANCE: invention refers to organic chemistry and pharmacology, namely to a novel compound used for therapy and prevention of metabolic syndrome. Disclosed (2S)-3-(4-{2-[4-(2-{[(1R,4aR,7S)-7-ethynyl-1,4a,7-trimethyl-1,2,3,4,4a,4b,5,6,7,8,10,10a-dodecahydrophenanthren-1-yl]formamido}ethoxy)phenyl]ethoxy}phenyl)-2-ethoxy-propanoic acid as an agent for therapy and prevention of metabolic syndrome.

EFFECT: using the invention provides effective therapy and prevention of metabolic syndrome.

1 cl, 10 dwg, 3 tbl, 2 ex

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RU 2 813 464 C1

Authors

Fomenko Vladislav Viktorovich

Khvostov Mikhail Vladimirovich

Blokhin Mikhail Evgenevich

Kuranov Sergei Olegovich

Luzina Olga Anatolevna

Salakhutdinov Nariman Faridovich

Dates

2024-02-12Published

2023-07-03Filed