NEW COMPOUND, METHOD OF ITS PREPARATION AND USE Russian patent published in 2024 - IPC C07C311/29 C07D207/27 C07D209/08 C07D209/14 C07D209/16 C07D209/86 C07D209/88 C07D211/10 C07D213/42 C07D231/56 C07D235/06 C07D235/14 C07D295/135 C07D401/04 C07D401/12 C07D417/12 C07D471/04 A61K31/18 A61P35/00 

Abstract RU 2814103 C1

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to a compound that inhibits Pin1 (peptidyl-prolyl-cis/trans isomerase interacting with NIMA 1), or a pharmaceutically acceptable salt thereof, a method of producing the said compound, a pharmaceutical composition containing as an active ingredient a compound that inhibits Pin1, and its use for the prevention or treatment of malignancy.

EFFECT: obtaining a new compound and a method of its preparation.

18 cl, 5 tbl, 185 ex

Similar patents RU2814103C1

Title Year Author Number
DIAMINOPYRIMIDINE DERIVATIVES AND METHODS FOR PRODUCTION THEREOF 2012
  • Lee Hyun-Joo
  • Kim Dong-Hoon
  • Kim Tae-Kyun
  • Yoon Young-Ae
  • Sim Jae-Young
  • Cha Myung-Hun
  • Jung Eun-Jung
  • Ahn Kyoung-Kyu
  • Lee Tai-Au
RU2587981C2
NOVEL DERIVATIVE OF PURINYLPYRIDINYLAMINO-2,4-DIFLUOROPHENYLSULPHONAMIDE, ITS PHARMACEUTICALLY ACCEPTABLE SALT, METHOD OF ITS OBTAINING AND PHARMACEUTICAL COMPOSITION, WHICH HAS INHIBITION ACTIVITY WITH RESPECT TO RAF-KINASE, CONTAINING CLAIMED COMPOUND AS ACTIVE INGREDIENT 2011
  • Shim Eun Kiong
  • Kim Nam Doo
  • Shim Tae Bo
  • Kim Seung Jong
RU2550038C2
COMPOUND INHIBITING FORMATION OF C-MYC/MAX/DNA COMPLEX 2017
  • Jeong, Kyung Chae
  • Lim, Hwan Jung
  • Park, Seong Jun
  • Seo, Ho Kyung
  • Ahn, Kyung Ohk
  • Lee, Sang Jin
  • Lee, Eun Sook
RU2727177C1
NEW PYRIMIDINE DERIVATIVE WITH AN EFFECT OF INHIBITING GROWTH OF CANCER CELLS AND PHARMACEUTICAL COMPOSITION CONTAINING IT 2018
  • Kim, Sung-Eun
  • Lee, Sunho
  • Rajesh, Rengasamy
  • Kang, Dae Ho
  • Ryu, Hyung Chul
  • Kim, Jae-Sun
  • Lee, Sangryul
  • Kim, Kyong Cheol
  • Rho, Jin Kyung
  • Lee, Jae Cheol
RU2744168C1
DIAMINOPYRIMIDINE DERIVATIVES AND METHODS FOR PRODUCTION THEREOF 2012
  • Lee Hyun-Joo
  • Kim Dong-Hoon
  • Kim Tae-Kyun
  • Yoon Young-Ae
  • Sim Jae-Young
  • Cha Myung-Hun
  • Jung Eun-Jung
  • Ahn Kyoung-Kyu
  • Lee Tai-Au
RU2587493C2
HETEROCYCLIC DERIVATIVES AND USE THEREOF 2014
  • Park Chan Khee
  • Li Sang Khvi
  • Im Dzunkhvan
  • Li Soon Ok
  • Kim Khoe Moon
  • Moon Sung Khyun
  • Kim Seungkhi
  • Kim Dzongmin
  • Ko Kvang Seok
  • Choi Bu Yang
  • Kim Byungkho
RU2681849C2
ANTICANCER PHARMACEUTICAL COMPOSITION 2017
  • Jeong, Kyung Chae
  • Lim, Hwan Jung
  • Park, Seong Jun
  • Seo, Ho Kyung
  • Ahn, Kyung Ohk
  • Lee, Sang Jin
  • Lee, Eun Sook
RU2724340C1
HETEROCYCLIC DERIVATIVES AND USE THEREOF 2015
  • Moon, Hyung Jo
  • Kim, Mi Sun
  • Kong, Minjung
  • Kim, Byungho
  • Ko, Kwang Seok
  • Kim, Jongmin
  • Lee, Soon Ok
  • Im, Junhwan
  • Lee, Sang Hwi
  • Park, Chan Hee
RU2734390C2
COMPOUND CONTAINING OXADIAZOLE AND A PHARMACEUTICAL COMPOSITION CONTAINING IT 2019
  • Ryu, Choon Ho
  • Han, Min Soo
  • Yoon, Yeo Jin
  • Kim, Yu Jin
  • Lee, Ka Eun
  • Lee, Ju Young
  • Jung, Myung Jin
  • Baek, Eun Hee
  • Shin, Yu Jin
  • Choi, Eun Ju
  • Kang, Young Soon
  • Kim, Yong Soo
  • Song, Yea Mi
  • Kim, Jin Sung
  • Lim, Hee Jeong
RU2789456C2
PYRIDOPYRIMIDINONE DERIVATIVES AND USE THEREOF AS AROMATIC HYDROCARBON RECEPTOR MODULATORS 2021
  • Song, Minsoo
  • Park, Ga Youn
  • Kang, Jihee
  • Lee, Eunhye
  • Park, Yoojin
  • Choi, Yujeong
  • Kim, Soong-Hyun
  • Ko, Eun Bi
  • Bae, Seri
  • Park, Jung-Sang
  • Cha, Daewon
  • Lee, Wonhyung
  • Joo, Min Sung
  • Yoon, Taeyoung
  • Doh, Hyounmie
  • Sung, Hyun Jung
  • Lee, Bo Ryeong
  • Kim, Yoonjung
RU2818954C1

RU 2 814 103 C1

Authors

Im, Chun Young

Min, Sang Hyun

Yu, Ji Hoon

Ko, Eun Bi

Kim, So Young

Lee, Seungyeon

Choi, Dong Kyu

Lee, Heejin

Park, Ga Young

Lee, Doohyun

Hong, Eunmi

Jeon, Hui-Jeon

Park, Young-Hoon

Han, Ye Ri

Kim, Nam Hui

Kim, Jun Woo

Oh, Bae Jun

Park, Jeong-Eun

Seo, Chang Hoon

Song, Minsoo

Ro, Seonggu

Shin, Dongkyu

Dates

2024-02-22Published

2021-01-15Filed