APPLICATION OF COMPOUND-AGONISTS OF HUMAN CB RECEPTOR FOR PREPARING MEDICINAL IMMUNOMODULATING AGENTS, NOVEL COMPOUNDS-AGONISTS OF CB RECEPTOR AND PHARMACEUTICAL COMPOSITIONS BASED ON THEREOF Russian patent published in 2003 - IPC

Abstract RU 2200736 C2

FIELD: medicine, organic chemistry. SUBSTANCE: invention proposes a novel agent with immunomodulating effect. Agent comprises selective agonist with affinity constant to CB2 receptor by at least 30 times lower than affinity constant to CB1 receptor. As such agonist the known or novel compounds can be used of general formulas (I) or (I') with radical values given in the invention claim. Except for immunomodulating effect, some compounds exhibit analgetic effect additionally. EFFECT: expanded arsenal of agents of prescription claimed. 13 cl, 1 test, 7 tbl, 11 sch, 13 ex

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RU 2 200 736 C2

Authors

Rinal'Di Mjuriel'

Bart Fransis

Kazellja P'Er

Kon'I Kristian

Ustrik Did'E

Bell Mal'Kol'M R.

D'Ambra Tomas E.

Filion Rishar E.

Dates

2003-03-20Published

1996-06-20Filed