FIELD: organic chemistry. SUBSTANCE: invention describes derivatives of N-sulfonyl-2- -oxoindole of the general formula (I) where values R1-R6 and m are given in point 1 of the invention. It describes also a method of their synthesis, intermediate substances and a pharmaceutical compositions based on compounds of the formula (I) showing affinity to vasopressin and/or oxytocin receptors. EFFECT: improved method of synthesis, affinity to receptors. 19 cl, 7 tbl, 211 ex
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