DERIVATIVES OF BENZOTHIEPINE-1,1-DIOXIDES, METHOD FOR THEIR PREPARING AND MEDICINAL AGENT Russian patent published in 2003 - IPC

Abstract RU 2220141 C2

FIELD: organic chemistry, chemical technology, pharmacy. SUBSTANCE: invention relates to derivatives of benzothiepine-1,1-dioxides and their additive salts with acids of the formula (I): wherein R1 means methyl, ethyl, propyl, butyl; R2 is hydrogen atom, OH; R3 is a saccharide residue being saccharide residue is mono- or multi-substituted if necessary with one or more protective group for saccharides; R4 means methyl, ethyl, propyl, butyl; R5 means methyl, ethyl, propyl, butyl; Z means (C=O)n-C1-C16-alkyl-NH-, covalent bond; n = 1. Compounds can be used as hypolipidemic agents. Invention describes also method for preparing these compounds and a medicinal agent based on thereof. EFFECT: improved preparing method, valuable medicinal properties of compounds. 13 cl, 1 tbl, 13 ex

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RU 2 220 141 C2

Authors

Frik Vendelin

Ehnzen Al'Fons

Glombik Khajner

Khojer Khubert

Dates

2003-12-27Published

1999-05-29Filed