DERIVATIVES OF TRIAZOLE OF AMIDE TYPE, PHARMACEUTICAL COMPOSITION BASED ON THEREOF AND METHOD FOR PROPHYLAXIS OR TREATMENT Russian patent published in 2004 - IPC

Abstract RU 2232761 C2

FIELD: organic chemistry, medicine, pharmacy.

SUBSTANCE: invention relates to derivatives of triazole of amide type or their pharmacologically acceptable salts of the formula (I):

wherein Ar1 represents phenyl group or similar group; Ar2 represents phenylene group or similar group; X represents sulfur atom or methylene group; R1 represents hydrogen atom or (C1-C3)-alkyl group; R2 represents hydrogen atom or (C1-C3)-alkyl group; R3 represents optionally substituted (C6-C10)-aryl group or similar group. Invention relates also to a pharmaceutical composition based on thereof eliciting anti-fungal effect and to method for prophylaxis or treatment of fungal infection. Invention provides preparing new compounds eliciting valuable pharmacological properties.

EFFECT: improved prophylaxis and treatment method, valuable medicinal properties of compounds.

22 cl, 2 tbl, 33 ex

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RU 2 232 761 C2

Authors

Utida Takuja

Konosu Tosijuki

Dates

2004-07-20Published

2001-03-27Filed