BENZOXEPIN PI3 INHIBITORS AND METHODS FOR USING THEM Russian patent published in 2015 - IPC C07D495/04 C07D495/14 C07D513/04 C07D513/14 A61K31/381 A61K31/429 A61K31/4365 A61P35/00 

Abstract RU 2557658 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to 2-(3-amino-1-(2,4-difluorophenyl)-1H-1,2,4-triazol-5-yl)-N-methyl-4,5-dihydrobenzo[b]thieno[2,3-d]oxepin-8-carboxamide. As well as to a pharmaceutical composition containing the above compound, to the use thereof and a set for treating.

EFFECT: 2-(3-amino-1-(2,4-difluorophenyl)-1H-1,2,4-triazol-5-yl)-N-methyl-4,5-dihydrobenzo[b]thieno[2,3-d]oxepin-8-carboxamide inhibiting PI3 kinase (PI3K).

6 cl, 15 dwg, 1 tbl, 610 ex

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RU 2 557 658 C2

Authors

Nikol' Blak'Er

Stiven Do

Dejnette Dadli

Adrian Dzh. Folks

Richard A. Goldsmit

Robert Khild

Tim Kheffron

Aleksandr Kolesnikov

Chudi Ndubaku

Alan G. Olivero

Stiven Prajs

Stiven Stejben

Bin'Tsin Vehj

Dates

2015-07-27Published

2010-09-27Filed