DERIVATIVES OF ARYL(OR HETEROARYL)AZOLYLCARBINOL FOR TREATMENT OF RESPIRATORY DISEASE Russian patent published in 2007 - IPC A61K31/381 A61K31/415 A61K31/4164 A61K31/551 A61K31/5517 A61P11/00 A61P11/06 A61P11/14 

Abstract RU 2294198 C2

FIELD: organic chemistry, medicine.

SUBSTANCE: invention proposes using aryl(or heteroaryl)azolylcarbinol of the general formula (I) wherein Ar means possibly substituted phenyl or thienyl; R means hydrogen atom or alkyl; R2 means dialkylaminoalkyl or azaheterocyclylalkyl; Het means unsubstituted azol of substituted with one or two substitutes, and their salts. Proposed derivatives can be used as an agent for treatment of chronic obstructive pulmonary diseases (cough, bronchitis, allergic rhinitis and asthma). Proposed compound depresses cough being without sedative effect.

EFFECT: valuable medicinal properties of compounds.

4 cl, 1 tbl, 3 ex

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RU 2 294 198 C2

Authors

Merse-Vidal Ramon

Andalus-Matero Blas

Frigola-Konstansa Khordi

Dates

2007-02-27Published

2002-03-21Filed