FIELD: organic chemistry, pharmaceuticals.
SUBSTANCE: invention relates to compounds of formula I , wherein substituents meanings are as defined in specification, and pharmaceutically acceptable salts or individual diastereomers thereof. Claimed compounds are useful as CGRP receptors antagonists in treatment or prophylaxis of headache, migraine, etc. Also disclosed are pharmaceutical compositions containing such compounds and uses thereof in treatment or prophylaxis of abovementioned diseases mediated by CGRP.
EFFECT: new CGRP receptor antagonists.
5 cl, 6 tbl, 40 ex
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Authors
Dates
2007-10-20—Published
2004-04-09—Filed