[4-(1-AMINOETHYL)CYCLOHEXYL]METHYLAMINE AND [6-(1-AMINOETHYL)TETRAHYDROPYRAN-3-YL]METHYLAMINE DERIVATIVES Russian patent published in 2014 - IPC C07D215/22 C07D407/06 C07D471/04 C07D491/04 C07D498/04 C07D513/04 A61K31/4709 A61K31/4375 A61P31/00 

Abstract RU 2515906 C2

FIELD: chemistry.

SUBSTANCE: invention relates to antibacterial compounds of formula (I), where R1 represents alkoxygroup; U, V and W each represents CH or one of U, V and W represents N, and each other represents CH; A represents CH2 or O; G represents CH=CH-E, where E represents phenyl group, mono- or di-substituted with halogen, or G represents group of one of the formulas given below , , where Z represents CH or N, Q represents O or S and K represents O or S; or salt of such compound. In addition, invention also relates to pharmaceutical composition based on formula (I) compound for prevention or treatment of bacterial infection, as well as to application of claimed compounds for obtaining medication for prevention or treatment of bacterial infection.

EFFECT: novel compounds, which can be applied in treatment of bacterial infection, are obtained and described.

23 cl, 1 tbl, 13 ex

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RU 2 515 906 C2

Authors

Kristian Khubshverlen

Georg Rjuehdi

Zhan-Filipp Sjurive

Kornelia Tsumbrunn-Aklin

Dates

2014-05-20Published

2009-06-02Filed