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IPC

C07D487/04(2006-01-01)

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Application

2006140602/04, 2006-11-16

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Start date

2006-11-16

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Actual filing date

2006-11-16

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Published

2007-12-10

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Inventor

Anisimova Vera AlekseevnaGalenko-Jaroshevskij Aleksandr PavlovichMinkin Vladimir IsaakovichTolpygin Ivan Evgen'EvichPorkhanova Anna VladimirovnaSergeev Vladimir VladimirovichVarlashkina Inessa AleksandrovnaFutorjanskaja Tamara NikolaevnaTlisheva Zarema ShumafovnaPelivanova Marija Kharlampievna

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Holder

Federal'Noe Gosudarstvennoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Federal'Nyj Universitet"Negosudarstvennoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Meditsinskij Institut"Federal'Noe Gosudarstvennoe Uchrezhdenie Nauchno-Tekhnicheskij Kompleks Glaza" Imeni Akademika S.N. Fedorova" Federal'Nogo Agentstva Po Zdravookhraneniju I Sotsial'Nomu Razvitiju Mntk Glaza" Im. Akad. S.N. Fedorova Roszdrava)

1-(3-PYRROLIDINOPROPYL)-2-(4-FLUOROPHENYL)IMIDAZO[1,2-a]-BENZIMIDAZOLE DIHYDROCHLORIDE POSSESSING TOPICAL ANESTHETIZING EFFECT Russian patent published in 2007 - IPC C07D487/04

Abstract RU 2312107 C1

FIELD: organic chemistry, medicine.

SUBSTANCE: invention relates to a novel 1,2-disubstituted derivative of imidazo[1,2-a]-benzimidazole. Invention describes 1-(3-pyrrolidinopropyl)-2-(4-fluorophenyl)imidazo[1,2-a]-benzimidazole dihydrochloride of the formula (I): Compound possesses topical anesthetizing effect in carrying out the surface (terminal) anesthesia. Invention provides preparing a novel compound possessing useful biological properties.

EFFECT: valuable medicinal property of compound.

3 tbl, 1 ex

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RU 2 312 107 C1

Authors

Anisimova Vera Alekseevna

Galenko-Jaroshevskij Aleksandr Pavlovich

Minkin Vladimir Isaakovich

Tolpygin Ivan Evgen'Evich

Porkhanova Anna Vladimirovna

Sergeev Vladimir Vladimirovich

Varlashkina Inessa Aleksandrovna

Futorjanskaja Tamara Nikolaevna

Tlisheva Zarema Shumafovna

Pelivanova Marija Kharlampievna

Dates

2007-12-10—Published

2006-11-16—Filed