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IPC

C07D487/04(2006-01-01)

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Application

2006140601/04, 2006-11-16

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Start date

2006-11-16

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Actual filing date

2006-11-16

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Published

2007-11-27

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Inventor

Anisimova Vera AlekseevnaGalenko-Jaroshevskij Aleksandr PavlovichMinkin Vladimir IsaakovichTolpygin Ivan Evgen'EvichVarlashkina Inessa AleksandrovnaTlisheva Zarema ShumafovnaLugovaja Irina Anatol'EvnaFutorjanskaja Tamara NikolaevnaUsov Aleksandr Valer'EvichZhukov Aleksej Vasil'Evich

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Holder

Federal'Noe Gosudarstvennoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Federal'Nyj Universitet"Negosudarstvennoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Meditsinskij Institut"Federal'Noe Gosudarstvennoe Uchrezhdenie Nauchno-Tekhnicheskij Kompleks Glaza" Imeni Akademika S.N. Fedorova" Federal'Nogo Agentstva Po Zdravookhraneniju I Sotsial'Nomu Razvitiju Mntk Glaza" Im. Akad. S.N.Fedorova Roszdrava)

1-(3-DIETHYLAMINOPROPYL)-2-(4-FLUOROPHENYL)-IMIDAZO[1,2-a]BENZIMIDAZOLE DIHYDROCHLORIDE ELICITING LOCAL ANESTHETIC EFFECT Russian patent published in 2007 - IPC C07D487/04

Abstract RU 2311416 C1

FIELD: organic chemistry, medicine.

SUBSTANCE: invention relates to a novel 1,2-disubstituted derivative of imidazo[1,2-a]imidazole. Invention describes 1-(3-diethylaminopropyl)-2-4-fluorophenyl)-imidazo[1,2-a]benzimidazole of the formula (I): . Compound elicits local anesthetic effect in surface (terminal), infiltration, conduction and epidural anesthesia. Invention provides synthesis of a novel compound possessing useful biological properties.

EFFECT: valuable medicinal properties of compounds.

6 tbl, 1 ex

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RU 2 311 416 C1

Authors

Anisimova Vera Alekseevna

Galenko-Jaroshevskij Aleksandr Pavlovich

Minkin Vladimir Isaakovich

Tolpygin Ivan Evgen'Evich

Varlashkina Inessa Aleksandrovna

Tlisheva Zarema Shumafovna

Lugovaja Irina Anatol'Evna

Futorjanskaja Tamara Nikolaevna

Usov Aleksandr Valer'Evich

Zhukov Aleksej Vasil'Evich

Dates

2007-11-27—Published

2006-11-16—Filed