1-(2-DIETHYLAMINOETHYL)-2-PHENYLIMIDAZO[1,2-A]BENZIMIDAZOLE DIHYDROCHLORIDE POSSESSING TOPICAL ANESTHETIC EFFECT AND PHARMACEUTICAL COMPOSITION BASED ON THEREOF Russian patent published in 2008 - IPC C07D487/04 A61K31/4188 

Abstract RU 2314312 C1

FIELD: organic chemistry, medicine.

SUBSTANCE: invention relates to a novel 1,2-disubstituted imidazo[1,2-a]benzimidazole. Invention describes 1-(2-diethylaminoethyl)-2-phenylimidazo[1,2-a]benzimidazole dihydrochloride of the formula (I): Also, invention describes a pharmaceutical composition with the topical anesthetic effect comprising 1-2-diethylaminoethyl)-2-phenylimidazo[1,2-a]benzimidazole dihydrochloride taken in the effective dose as an active component. Invention provides synthesis of a novel compound possessing valuable biological properties.

EFFECT: valuable medicinal properties of compound and pharmaceutical composition.

2 cl, 6 tbl, 1 ex

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Authors

Anisimova Vera Alekseevna

Galenko-Jaroshevskij Aleksandr Pavlovich

Minkin Vladimir Isaakovich

Tolpygin Ivan Evgen'Evich

Spasov Aleksandr Alekseevich

Varlashkina Inessa Aleksandrovna

Piskunov Aleksandr Valerievich

Lugovaja Irina Anatol'Evna

Futorjanskaja Tamara Nikolaevna

Dates

2008-01-10Published

2006-11-16Filed